2. Signaling Pathways
  3. Vitamin D Related/Nuclear Receptor
  4. Estrogen Receptor/ERR
  5. ERRγ Isoform
  6. ERRγ Inhibitor

ERRγ Inhibitor

ERRγ Inhibitor (1):

Cat. No. Product Name Effect Purity
  • HY-111226
    GSK5182
    		Inhibitor 99.85%
    GSK5182 is a highly selective and orally active inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM. GSK5182 does not interact with other nuclear receptors, including ERRα or ERα. GSK5182 also induces reactive oxyen species (ROS) generation in hepatocellular carcinoma (HCC).